6-ethyl-7-hydroxy-4-methylchromen-2-one;化合物T42046-ethyl-7-hydroxy-4-methylcoumarin;6-ethyl-7-hydroxy (2024/9/8)
簡介:6-ethyl-7-hydroxy-4-methylchromen-2-one is a fluorescent dye.
Delamanid德拉馬尼迪拉馬尼|||德拉馬尼|||OPC-67683 (2024/9/8)
簡介:delamanid (opc-67683) is an anti-tuberculosis agent derived from the nitro-dihydro-imidazooxazole class of compounds that inhibits mycolic acid synthesis of bacterial cell wall.
Avibactam sodium;阿維巴坦鈉AVE-1330A|||NXL-104;阿維巴坦|||AVE-1330A|||阿維巴坦鈉|||NXL-104 (2024/9/8)
簡介:avibactam sodium (nxl-104) is a reversible β-lactamase inhibitor (ic50: 8/80/38 nm, for tem-1/p99/kpc-2 β-lactamases).
Sacubitril hemicalcium salt;LCZ696中間體AHU-377 (hemicalcium salt)|||AHU377 calcium salt;AHU-377 (hemic (2024/9/8)
簡介:sacubitril hemicalcium salt (ahu377 calcium salt) is a potent nep inhibitor with an ic50 of 5 nm. sacubitril hemicalcium salt is a component of the heart failure medicine lcz696. sacubitril hemicalcium salt is a prodrug of lbq657, which is an inhibitor of the zinc metallopeptidase neprilysin. neprilysin degrades a variety of vasoactive peptides such as atrial and brain natriuretic peptide, bradykinin, adrenomedullin, and endothelin-1. inhibition of neprilysin leads to an increased level of these
Desmethyl-VS-5584;化合物Desmethyl-VS-5584Desmethyl-VS-5584 (2024/9/8)
簡介:desmethyl-vs-5584 is a dimethyl analog of vs-5584, which is a novel and highly selective pi3k/mtor kinase inhibitor for the treatment of cancer.
T.cruzi-IN-1;T.cruzi InhibitorMDK1088|||T.cruzi Inhibitor;MDK1088|||T.cruzi Inhibitor (2024/9/8)
簡介:t.cruzi-in-1 (mdk1088) is a trypanosoma cruzi inhibitor.
HZ-1157;化合物HZ1157HZ1157|||DHFR-inhibitor;HZ1157|||DHFR-inhibitor (2024/9/8)
簡介:hz-1157 (dhfr-inhibitor) is a hepatitis c virus (hcv) inhibitor with inhibitory activities toward hcv ns3/4a protease.
Betahistine EP Impurity C;化合物NSC19005NSC19005;NSC19005 (2024/9/8)
簡介:betahistine ep impurity c (nsc19005) is structurally related to betahistine. betahistine ep impurity c is a dimer of betahistine.
Betahistine;倍他司汀PT 9 base|||Vasomotal|||Serc base;PT 9 base|||倍他司汀|||Vasomotal|||Serc base (2024/9/8)
簡介:betahistine (vasomotal) is a histamine analog and h1 receptor agonist that serves as a vasodilator. it is used in meniere disease and in vascular headaches but may exacerbate bronchial asthma and peptic ulcers. betahistine dihydrochloride is an anti-vertigo drug. it is commonly prescribed for balance disorders or to alleviate vertigo symptoms associated with ménière´s disease.
Raf inhibitor 2;化合物CID25014542CID-25014542|||CID 25014542|||CID25014542;CID-25014542|||CID 25014542| (2024/9/8)
簡介:raf inhibitor 2 (cid 25014542) is novel inhibitor of raf kinases.
TD-198946;化合物TD198946TD198946|||TD 198946;TD198946|||TD 198946 (2024/9/8)
簡介:td-198946, a potent chondrogenic agent, is a thienoindazole derivative.
hnps-PLA Inhibitor;化合物hnps-PLA Inhibitorhnps-PLA Inhibitor (2024/9/8)
簡介:hnps-pla inhibitor is an inhibitor of human nonpancreatic secretory phospholipase a (hnps-pla).
Multi-kinase inhibitor 1;化合物Multi-kinase inhibitor IMulti-kinase inhibitor I;Multi-kinase inhibitor (2024/9/8)
簡介:multi-kinase inhibitor 1 (multi-kinase inhibitor i) is a multi-kinase inhibitor.
Ticlopidine;噻氯匹定PCR 5332|||Ticlid;PCR 5332|||Ticlid|||噻氯匹定 (2024/9/8)
簡介:ticlopidine (pcr 5332) is an antiplatelet drug in the thienopyridine family which is an adenosine diphosphate (adp) receptor inhibitor.
4-Oxofenretinide;4-氧代維甲酰酚胺3-Keto fenretinide;3-Keto fenretinide|||4-氧代維甲酰酚胺 (2024/9/8)
簡介:4-oxofenretinide (3-keto fenretinide) , a recently identified fenretinide metabolite, induces marked g2-m cell cycle arrest and apoptosis.
SDZ285428化合物SDZ285-428SDZ285-428 (2024/9/8)
簡介:sdz285428 is a cyp24a1 inhibitor.
Gemcitabine monophosphate sodium salt hydrate;吉西他濱單磷酸酯Gemcitabine monophosphate sodium salt hydrate (2024/9/8)
簡介:gemcitabine monophosphate disodium salt is a monophosphate derivative of gemcitabine.
AC-264613;化合物AC264613AC264613;AC264613 (2024/9/8)
簡介:ac-264613 is an agonist of the gpcr protease-activated receptor 2 (par2). ac-264613(ac264613) suppresses interferon regulatory factor 5 and decreases interleukin-12p40 production by lipopolysaccharide-stimulated macrophages. ac-264613(ac264613) activated par2 signaling in cellular proliferation assays, phosphatidylinositol hydrolysis assays, and ca(2+) mobilization assays, with potencies ranging from 30 to 100 nm.
lavendustin C;N-(2,5-二羥基芐基)-5-氨基水楊酸HDBA|||NSC 666251;HDBA|||NSC 666251|||N-(2,5-二羥基芐基)-5-氨基水楊酸 (2024/9/8)
簡介:lavendustin c (nsc 666251) is a potent inhibitor of epidermal growth factor (egf) receptor-associated tyrosine kinase.
NSC 409012;5-(4-碘苯亞甲基)羅丹寧5-(4-iodobenzylidene)rhodanine;5-(4-iodobenzylidene)rhodanine|||5-(4-碘苯亞甲基) (2024/9/8)
簡介:nsc-409012 (5-(4-iodobenzylidene)rhodanine) is an active compound that has been found to have a variety of biochemical and physiological effects, including regulation of gene expression, cell proliferation and apoptosis. it also possesses anti-inflammatory, anti-tumor, antioxidant and antifungal activities.
lavendustin A;薰草菌素RG-14355|||NSC 678027;RG-14355|||NSC 678027|||薰草菌素 (2024/9/8)
簡介:lavendustin a (rg-14355) is a potent, cell-permeable inhibitor of epidermal growth factor receptor (egfr) tyrosine kinase.
lavendustin B薰草菌素B薰草菌素B (2024/9/8)
簡介:lavendustin b is a tyrosine kinase inhibitor and an inhibitor of hiv-1 integrase (in) interaction with its cognate cellular cofactor, lens epithelium-derived growth factor (ledgf/p75).
Cosan 528;化合物Cosan 528Cosan 528 (2024/9/8)
簡介:cosan-528 is a bioactive chemical.
Adipamidoxime;化合物AdipamidoximeNSC70868;NSC70868 (2024/9/8)
簡介:adipamidoxime (nsc-70868) is an oxime-active compound that inhibits the growth of certain bacteria, fungi, and viruses and has some anti-inflammatory and anti-tumor activities.
Probucol disuccinate;普羅布考Probucol disuccinate (2024/9/8)
簡介:probucol is an anti-hyperlipidemic drug initially developed in the treatment of coronary artery disease by lowering the level of cholesterol in the bloodstream by increasing the rate of ldl catabolism.
NSC 80538;化合物NSC 80538NSC 80538 (2024/9/8)
簡介:nsc 80538 is an inhibitor of mek kinase pb1 domains in multiplex hts assays.
U 19963;化合物U 19963U 19963 (2024/9/8)
簡介:u 19963 is a potent inhibitor of several enzymes and receptors and has been used to study the effects of drugs on biological systems. it has been found to possess a wide range of biological activities, including anti-inflammatory, anti-tumor and antibacterial properties.
rac-BHFF;化合物rac-BHFF(R,S)-BHFF;(R,S)-BHFF (2024/9/8)
簡介:rac-bhff ((r,s)-bhff) is potent and selective gaba b receptor positive allosteric modulator that increases the potency and efficacy of gaba ( > 15-fold and > 149% respectively). it exhibits anxiolytic activity in vivo and is orally active.
Loflucarban;氯氟卡班Fluonilid;氯氟卡班|||Fluonilid (2024/9/8)
簡介:loflucarban (fluonilid) is an antimycotic compoud.
NSC 191412;化合物NSC 191412NSC 191412 (2024/9/8)
簡介:nsc 191412 interacts with a variety of enzymes and receptors, including acetylcholinesterase and receptors for the neurotransmitter dopamine, and is an agonist or activator of these enzymes and receptors.