9月
JNJ-47965567；化合物JNJ-47965567JNJ-479655；JNJ-479655 (2024/9/8)
簡(jiǎn)介：jnj-47965567 (jnj-479655) is a selective antagonist of the purinergic receptor p2x subtype 7 (p2x7), a ligand-gated ion channel(with pkis of 7.9 and 8.7 for human and rat p2x7, respectively).
Flibanserin；氟立班絲氨BIMT-17BS|||Girosa|||BIMT-17；BIMT-17BS|||氟立班絲氨|||Girosa|||BIMT-17 (2024/9/8)
簡(jiǎn)介：flibanserin (girosa) is a serotonergic antidepressant used to treat hypoactive sexual desire disorder. flibanserin has been associated with a low rate of minor serum aminotransferase elevations during treatment but has not been linked to instances of clinically apparent acute liver injury.
MTX-211；化合物MTX211MTX 211；MTX 211 (2024/9/8)
簡(jiǎn)介：mtx-211, an inhibitor of egfr and pi3k, is used for the therapy of cancer and other diseases.
(R)-GNE-140；化合物(R)-GNE-140GNE-140；GNE-140 (2024/9/8)
簡(jiǎn)介：(r)-gne-140 (gne-140) is an effective ldha/ldhb inhibitor (ic50s: 3/5 nm) and is 18-fold more potent than s enantiomer.
NS 11021；化合物NS11021NS11021；NS11021 (2024/9/8)
簡(jiǎn)介：ns 11021 (ns11021) , a novel opener of large-conductance ca(2+)-activated k(+) channels
THZ531；化合物THZ531THZ531 (2024/9/8)
簡(jiǎn)介：thz531 is a covalent inhibitor of both cdk12(ic50=158 nm) and cdk13(ic50=69 nm).
ThiaprolineL-硫代脯氨酸L-Thioproline|||L-Thiaproline|||L-硫代脯氨酸 (2024/9/8)
簡(jiǎn)介：thiaproline (l-thiaproline) has been used in peptide coupling reactions.
(+)-Isocorydine hydrochloride；鹽酸異可利定Isocorydine HCl；鹽酸異可利定|||Isocorydine HCl (2024/9/8)
簡(jiǎn)介：(+)-isocorydine hydrochloride (isocorydine hcl) is a eukaryote protein kinases inhibitor.
Preladenant；瑞德南特SCH-420814；SCH-420814|||瑞德南特 (2024/9/8)
簡(jiǎn)介：preladenant (sch-420814) is an orally bioavailable antagonist of the adenosine a2a receptor (ki: 1.1 nm) and has >1000-fold selectivity over all other adenosine receptors.
Mc-?Val-?Ala-?PAB；化合物Mc-Val-Ala-PABMc-Val-Ala-PAB；Mc-Val-Ala-PAB (2024/9/8)
簡(jiǎn)介：mc-val-ala-pab, an effective linker, is utilized in antibody-drug-conjugate (adc).
hVEGF-IN-1；化合物hVEGF-IN-1hVEGF-IN-1 (2024/9/8)
簡(jiǎn)介：hvegf-in-1 inhibits human vegf-a translation and has antitumor activity.
Succinobucol；化合物SuccinobucolProbucol monosuccinate|||AGI-1067；Probucol monosuccinate|||AGI-1067 (2024/9/8)
簡(jiǎn)介：succinobucol (probucol monosuccinate) is a novel phenolic antioxidant small molecule with anti-oxidant and anti-inflammatory properties. it designed to treat atherosclerosis of the blood vessels of the heart or coronary artery disease.
Fmoc-Val-Ala-PAB-OH；化合物Fmoc-Val-Ala-PABFmoc-Val-Ala-PAB；Fmoc-Val-Ala-PAB (2024/9/8)
簡(jiǎn)介：fmoc-val-ala-pab-oh (fmoc-val-ala-pab) is a useful linker for making antibody-drug-conjugation (adc) conjugate for targeting drug delivery. it is also utilized in the synthesis of rgd peptidomimetic-paclitaxel conjugates bearing lysosomally cleavable linkers.
Crisaborole；克立硼羅AN-2728|||PF-06930164；克立硼羅|||AN-2728|||PF-06930164 (2024/9/8)
簡(jiǎn)介：crisaborole (an-2728) is a phosphodiesterase 4 inhibitor.
Levamlodipine besylate；左旋氨氯地平(S)-Amlodipine Besylate (103129-82-4(free base))；左旋氨氯地平|||(S)-Amlodipin (2024/9/8)
簡(jiǎn)介：levamlodipine besylate ((s)-amlodipine besylate (103129-82-4(free base))) , also known as s-amlodipine, is a pharmacologically active enantiomer of amlodipine, an antihypertensive and anti-anginal medication. levamlodipine besylate belongs to the dihydropyridine group of calcium channel blockers. the names s-amlodipine and levamlodipine may be used interchangeably as both substances are the same, however, with differing nomenclature. as a racemic mixture, amlodipine contains (r) and (s)-amlodipi
SRI-011381；化合物SRI011381SRI-011381 (2024/9/8)
簡(jiǎn)介：sri-011381, a new-type agonist of the tgf-beta signaling pathway, is utilized in the treatment of alzheimer´s disease.
S-methyl-KE-298；化合物S-methyl-KE-298S-methyl-KE-298 (2024/9/8)
簡(jiǎn)介：s-methyl-ke-298 is the second main metabolite in plasma,is a methyl conjugate of deacetyl-ke-298.ke-298 inhibits matrix metalloproteinase (mmp-1) production from ?rheumatoid arthritis (ra) synovial cells.
Endoxifen；N-去甲基-4-羥基-(E/Z)-N-desmethyl-4-hydroxy Tamoxifen|||(E/Z)-Endoxifen；(E/Z)-N-desmethyl-4-hyd (2024/9/8)
簡(jiǎn)介：(e/z)-endoxifen ((e/z)-endoxifen) is an active metabolite of tamoxifen produced by the sequential action of cytochrome p450 (cyp) isoforms, including cyp2d6. it is a strong anti-estrogen, as it has an approximately 100-fold greater affinity for estrogen receptors than tamoxifen. as the efficient conversion of tamoxifen to endoxifen depends on cyp2d6, polymorphisms in this cyp isoform can impact the effectiveness of tmx treatment.
Gcase activator 1；化合物L(fēng)TI291LTI-291|||LTI 291|||LTI291；LTI-291|||LTI 291|||LTI291 (2024/9/8)
簡(jiǎn)介：gcase activator 1 (lti-291) is a glucocerebrosidase (gcase) activator.
Esonarimod；化合物EsonarimodKE-298；KE-298 (2024/9/8)
簡(jiǎn)介：esonarimod (ke-298) is an antirheumatic drug.
Hydroxyfasudil；羥基法舒地爾Hydroxy-Fasudil|||HA-1100；Hydroxy-Fasudil|||HA-1100|||羥基法舒地爾 (2024/9/8)
簡(jiǎn)介：hydroxyfasudil (hydroxy-fasudil) is a rock inhibitor(ic50s of 0.73 and 0.72 μm for rock1 and rock2, respectively).
Hydroxyfasudil Hydrochloride羥基法舒地爾鹽酸鹽Hydroxyfasudil (HA-1100) HCl|||羥基法舒地爾鹽酸鹽|||RHO-激酶抑制劑|||HA 1100 (2024/9/8)
簡(jiǎn)介：hydroxyfasudil hydrochloride (ha 1100 hydrochloride) is a rock1/2 inhibitor (ic50s: 0.73/0.72 μm).
Fluanisone；氟苯丙酮哌嗪Sedalande|||Haloanison；Sedalande|||氟苯丙酮哌嗪|||Haloanison (2024/9/8)
簡(jiǎn)介：fluanisone (haloanison) is a butyrophenone derivative with sedative properties. it is a typical antipsychotic and is used in the treatment of schizophrenia.
Melitracen hydrochloride；鹽酸美力他欣Thymeol hydrochloride|||Melixeran；鹽酸美利曲辛|||鹽酸美力他欣|||Thymeol hydrochlo (2024/9/8)
簡(jiǎn)介：melitracen hydrochloride (thymeol hydrochloride) , an antidepressant, is used as potential dopamine d1/2 receptor antagonist to treat depression.
Furagin呋喃烯啶F-35|||Akritoin|||Furazidine|||NF-416|||呋喃烯啶|||Furazidin (2024/9/8)
簡(jiǎn)介：furagin (furazidine) is a nitrofuran derivative with anti-infective activity used for urinary tract infections.
4-Hydroxyquinoline；4-羥基喹啉4-Quinolinol|||Quinolin-4-Ol；4-羥基喹啉|||4-Quinolinol|||Quinolin-4-Ol (2024/9/8)
簡(jiǎn)介：4-hydroxyquinoline (4-quinolinol) is a hydroxylated quinoline derivative with antimicrobial activity. it shows growth-inhibitory effects against intestinal bacteria. it also can be used as sacrificial scavengers of the photogenerated oxygen species.
Diroximel fumarate；化合物Diroximel FumareteDiroximel Fumarete；Diroximel Fumarete (2024/9/8)
簡(jiǎn)介：diroximel fumarate (diroximel fumarete), a prodrug of monomethyl fumarate in a controlled-release formulation, rapidly and potently converts to mmf in the body.
Cefquinome sulfate硫酸頭孢喹肟硫酸頭孢喹肟|||硫酸頭孢喹諾 (2024/9/8)
簡(jiǎn)介：cefquinome sulfate is a semisynthetic, broad-spectrum, fourth-generation aminothiazolyl cephalosporin with antibacterial activity.
Buparvaquone布帕伐醌布帕伐醌|||Butalex|||BW 720C (2024/9/8)
簡(jiǎn)介：buparvaquone (bw 720c) is a hydroxynaphthoquinone antiprotozoal drug related to atovaquone and parvaquone.
CHMFL-BMX-078；化合物CHMFL-BMX-078CHMFL-BMX-078 (2024/9/8)
簡(jiǎn)介：chmfl-bmx-078 is a highly potent and selective type ii irreversible bmx kinase inhibitor with an ic50 of 11 nm.
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