9月
Picropodophyllotoxin；苦鬼臼毒素AXL 1717|||Picropodophyllin；AXL 1717|||Picropodophyllin|||苦鬼臼毒素 (2024/9/8)
簡(jiǎn)介：picropodophyllotoxin (axl 1717) is a cyclolignan alkaloid found in the mayapple plant family (podophyllum peltatum), and a small molecule inhibitor of the insulin-like growth factor 1 receptor (igf1r) with potential antineoplastic activity. picropodophyllotoxin (axl 1717) specifically inhibits the activity and downregulates the cellular expression of igf1r without interfering with activities of other growth factor receptors, such as receptors for insulin, epidermal growth factor, platelet-derive
Ethyl trans-caffeate；咖啡酸乙酯Ethyl caffeate|||Caffeic Acid Ethyl Ester；咖啡酸乙酯|||Ethyl caffeate|||Caffeic (2024/9/8)
簡(jiǎn)介：1. ethyl trans-caffeate (caffeic acid ethyl ester) has anti-inflammatory activity. 2. ethyl trans-caffeate may as a promising natural compound for future application in chronic liver disease. 3. ethyl trans-caffeate is a potent chemopreventive compound against skin carcinogenesis caused by solar uv exposure. 4. ethyl trans-caffeate is the high-resolution structures of representative inhibitors in complex with human pancreatic α-amylase. 5. ethyl trans-caffeate strongly inhibits neoplastic transf
coniferyl ferulate；阿魏酸松柏酯coniferyl ferulate (2024/9/8)
簡(jiǎn)介：coniferyl ferulate is a strong inhibitor of glutathione s-transferase (gst) isolated from radix angelicae sinensis. it shows strong inhibition of human placental gst (ic50: 0.3 μm). it also reverses multidrug resistance and downregulates p-glycoprotein.
(E)-Ferulic acid methyl ester；(E)-阿魏酸甲酯Methyl ferulate|||Methyl (E)-ferulate；Methyl ferulate|||Methy (2024/9/8)
簡(jiǎn)介：(e)-ferulic acid methyl ester (methyl (e)-ferulate) is a possible inhibitor of the mitogen activated phosphor kinase pathway, it could be a potential anti-inflammatory agent isolated for the first time in medicinal plant s. tuberosa. (e)-ferulic acid methyl ester has promising anthelmintic activity against haemonchus contortus.
α-Linolenic acid；α-亞麻酸Alpha-Linolenic Acid|||Linolenic acid；Alpha-Linolenic Acid|||Linolenic acid||| (2024/9/8)
簡(jiǎn)介：α-linolenic acid (alpha-linolenic acid) is an essential fatty acid belonging to the omega-3 fatty acids group. it is highly concentrated in certain plant oils and has been reported to inhibit the synthesis of prostaglandin resulting in reduced inflammation and prevention of certain chronic diseases.
Chamigrenal；恰米醛Chamigrenal (2024/9/8)
簡(jiǎn)介：β-chamigrenal has anti-inflammatory activity, it has inhibitory effects on lipopolysaccharide-induced nitric oxide and prostaglandin e2 production in raw 264.7 macrophages. chamigrenal shows platelet-activating factor antagonistic activity and the ic(50) value of 1.2x10(-4) m; it also exhibits weak cytotoxicity towards mcf-7 cells(ic50=30.50 um).
Vitamin B6維生素B6維生素B6 (2024/9/8)
簡(jiǎn)介：vitamin b6 is a component of some coenzymes in human body, which is involved in a variety of metabolic reactions, especially related to amino acid metabolism.clinical application of vitamin b6 in the prevention and treatment of pregnancy and radiation sickness vomiting.
L-LeucineL-亮氨酸(S)-Leucine|||Leu|||L-亮氨酸|||亮氨酸 (2024/9/8)
簡(jiǎn)介：l-leucine ((s)-leucine) is one of nine essential amino acids in humans (provided by food), l-leucine is important for protein synthesis and many metabolic functions. l-leucine contributes to regulation of blood-sugar levels; growth and repair of muscle and bone tissue; growth hormone production; and wound healing. l-leucine also prevents breakdown of muscle proteins after trauma or severe stress and may be beneficial for individuals with phenylketonuria. l-leucine is available in many foods and
Bronze Red；808猩紅Scarlet 808；808猩紅|||Scarlet 808 (2024/9/8)
簡(jiǎn)介：bronze red, an amide class organic compound, is utilized for content determination, identification, and pharmacological experiments.
Allocryptopine；別隱品堿Thalictrimine|||Fagarine I；Thalictrimine|||Fagarine I|||別隱品堿 (2024/9/8)
簡(jiǎn)介：allocryptopine (thalictrimine) induces muscle contraction and relaxation in urinary bladder and ileum, respectively.
Manninotriose；甘露三糖Manninotriose (2024/9/8)
簡(jiǎn)介：manninotriose is the main carbohydrate of ono sesame (lamium. lamiaceae), participates in rfo metabolism and may play an important role.
IACS-15414；IACS-15414IACS-15414 (2024/9/8)
簡(jiǎn)介：iacs-15414 is a potent shp2 inhibitor that is effective when administered orally, demonstrating an ic50 value of 122 nm.
BET bromodomain inhibitor 1；BET bromodomain inhibitor 1BET bromodomain inhibitor 1 (2024/9/8)
簡(jiǎn)介：bet bromodomain inhibitor 1 is an orally active, selective inhibitor of bromodomain and extra-terminal (bet) proteins. it specifically inhibits brd4 with an ic50 of 2.6 nm. additionally, bet bromodomain inhibitor 1 demonstrates high affinities towards brd2(2), brd3(2), brd4(1), brd4(2), and brdt(2) with kd values of 1.3 nm, 1.0 nm, 3.0 nm, 1.6 nm, and 2.1 nm, respectively. this compound exhibits anti-cancer activity.
PROTAC CDK9 ligand-1；PROTAC CDK9 ligand-1PROTAC CDK9 ligand-1；PROTAC CDK9 ligand-1 (2024/9/8)
簡(jiǎn)介：protac cdk9 ligand-1 is a cdk9 ligand that can be used in the synthesis of protacs.
PROTAC CDK9 degrader-4；PROTAC CDK9 degrader-4PROTAC CDK9 degrader-4；PROTAC CDK9 degrader-4 (2024/9/8)
簡(jiǎn)介：protac cdk9 degrader-4 is a potent and efficacious chemical compound designed specifically to degrade cdk9, a protein involved in transcription regulation. this compound effectively targets and reduces the levels of cdk9, thereby modulating transcriptional activity.
TRV120055；TRV120055TRV120055；TRV120055 (2024/9/8)
簡(jiǎn)介：trv120055, a gq-biased agonist, demonstrates a 10-fold higher molecular efficacy when tested against the at1r-gq fusion protein in comparison to the at1r-βarr2 fusion protein.
Sovilnesib；化合物SovilnesibAMG650；AMG650 (2024/9/8)
簡(jiǎn)介：sovilnesib is a kinesin-like protein kif18a inhibitor. sovilnesib can be used for the cancer research.
PRMT5-IN-15PRMT5-IN-15PRMT5-IN-15 (2024/9/8)
簡(jiǎn)介：prmt5-in-15 is a prmt5 inhibitor with an ic 50 value of 0.84 nm.
FGFR1 inhibitor-2FGFR1 inhibitor-2FGFR1 inhibitor-2 (2024/9/8)
簡(jiǎn)介：fgfr1 inhibitor-2 (with an ic50 of 4.55 μm in mda-mb-231 cells) is a potent inhibitor of fgfr1. it is specifically useful for studying metastatic triple-negative breast cancer.
18-Oxocortisol；18-Oxocortisol18-Oxocortisol (2024/9/8)
簡(jiǎn)介：18-oxocortisol is a cortisol derivative generated by aldosterone synthase (cyp11b2). it acts as a naturally occurring mineralocorticoid agonist and serves as a biomarker in adrenal vein sampling.
HDAC-IN-26；HDAC-IN-26HDAC-IN-26 (2024/9/8)
簡(jiǎn)介：hdac-in-26 is a highly selective class i hdac inhibitor with an ec 50 value of 4.7 nm.
D(+)-Galactosamine hydrochlorideD-氨基半乳糖鹽酸鹽D-半乳糖胺鹽酸鹽|||D-氨基半乳糖鹽酸鹽|||D-Galactosamine HCl (2024/9/8)
簡(jiǎn)介：d(+)-galactosamine hydrochloride (d-galactosamine hcl) hepatotoxicity is associated with endotoxin sensitivity and mediated by lymphoreticular cells in mice.
JQKD82 trihydrochloride；三鹽酸JQKD82JQKD82 trihydrochloride (2024/9/8)
簡(jiǎn)介：jqkd82 trihydrochloride, a cell-permeable and selective inhibitor of kdm5, enhances h3k4me3 levels and is utilized in multiple myeloma research.
壓電雨量計(jì) (2024/9/8)
簡(jiǎn)介：壓電雨量計(jì)，廣泛應(yīng)用于氣象環(huán)境監(jiān)測(cè)、水文水利綜合監(jiān)測(cè)站、交通道路監(jiān)測(cè)、農(nóng)林、風(fēng)力發(fā)電等有關(guān)部門用來(lái)遙測(cè)降水量、降水強(qiáng)度、降水起止時(shí)間。用于防洪、供水調(diào)度、電站水庫(kù)水情管理為目的水文自動(dòng)測(cè)報(bào)系統(tǒng)、自動(dòng)野外測(cè)報(bào)站等。
JQKD82；化合物JQKD82JADA82|||PCK82|||JQKD82；JADA82|||PCK82|||JQKD82 (2024/9/8)
簡(jiǎn)介：jqkd82 is a selective inhibitor of kdm5 and increases h3k4me3. jqkd82 can be used in studies about the treatment of multiple myeloma.
BOC-NH-PEG2-propene；BOC-NH-PEG2-propeneBOC-NH-PEG2-propene；BOC-NH-PEG2-propene (2024/9/8)
簡(jiǎn)介：boc-nh-peg2-propene is a peg-based linker for protacs which joins two essential ligands, crucial for forming protac molecules. this linker enables selective protein degradation by leveraging the ubiquitin-proteasome system within cells.
LOX-IN-3 dihydrochloride；化合物L(fēng)OX-IN-3 dihydrochlorideLOX-IN-3 dihydrochloride (2024/9/8)
簡(jiǎn)介：lox-in-3 dihydrochloride is an inhibitor of lysyl oxidase (lox). lox-in-3 dihydrochloride inhibited bovine lox (ic50<10 μm) and human loxl2 (ic50<1 μm)activities.
(S,R,S)-AHPC-Me-CO-CH2-PEG3-NH2(S,R,S)-AHPC-Me-CO-CH2-PEG3-NH2(S,R,S)-AHPC-Me-CO-CH2-PEG3-NH2 (2024/9/8)
簡(jiǎn)介：(s,r,s)-ahpc-me-co-ch2-peg3-nh2 is a synthetic e3 ligase ligand-linker conjugate comprised of a vhl ligand and a linker. it is utilized in protac brd4 degrader-5 and protac brd4 degrader-5-co-peg3-n3.
上海高空蜘蛛人外墻維修 (2024/9/8)
簡(jiǎn)介：高空
PKM2-IN-3PKM2-IN-3PKM2-IN-3 (2024/9/8)
簡(jiǎn)介：pkm2-in-3 is a potent pkm2 kinase inhibitor, displaying an ic 50 value of 4.1 μm. the compound effectively suppresses pkm2-mediated glycolysis and nlrp3 activation, thereby exerting an anti-neuroinflammatory effect.
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