Ellipticine hydrochloride;玫瑰樹堿鹽酸鹽Ellipticine HCl|||NSC 71795 (hydrochloride);Ellipticine HCl|||NSC 7 (2024/9/8)
簡介:ellipticine hydrochloride (nsc-71795 (hydrochloride)) is a potent antineoplastic agent; inhibits dna topoisomerase ii activities.
Arg-Gly-Asp TFA (99896-85-2(free base));化合物Arg-Gly-Asp TFARGD Trifluoroacetate|||RGD;RGD Trifluoroac (2024/9/8)
簡介:arg-gly-asp tfa (99896-85-2(free base)) (rgd trifluoroacetate) is a tripeptide that effectively triggers cell adhesion, addresses certain cell lines and elicits specific cell responses; binds to integrins.
NS309;化合物NS309NS309 (2024/9/8)
簡介:ns309 is a nonselective activator of small- and intermediate-conductance ca2+-activated k+ (sk/kca2 and ik/kca3.1) channels (ec50s range from 0.12-1.2 μm for sk channels and 10-90 nm for ik channels). it can also activate voltage-gated kv11.1 channels (herg; ic50 = 1 μm), but does not, however, affect large conductance (bk/kca1.1) channels. ns309 can modulate neuronal firing patterns by enhancing sk-mediated hyperpolarizing effects. it is 730-fold (sk channels) and 7,400-fold (ik channels) more
EN300-203561;化合物EN300-203561EN300-203561 (2024/9/8)
簡介:en300-203561 has a wide range of applications in life science related research.
Exo1;化合物Exo1Exo1 (2024/9/8)
簡介:exo1 is an inhibitor of the exocytic pathway
PDM2;化合物PDM2PDM2 (2024/9/8)
簡介:pdm 2 is a potent and selective aryl hydrocarbon receptor (ahr) antagonist.
CAY 10465;化合物CAY10465CAY10465|||CAY10465 Exclusive;CAY10465|||CAY10465 Exclusive (2024/9/8)
簡介:cay 10465 is a selective and high-affinity ahr agonist, with a ki of 0.2 nm, and shows no effect on estrogen receptor (ki >100000 nm).
2119738-71-3;化合物2119738-71-32119738-71-3 (2024/9/8)
簡介:compound 2119738-71-3 interacts with the fak receptor.
NT157;化合物NT157NT157 (2024/9/8)
簡介:nt157 is a small molecule tyrphostin targeting irs protein and has the potential to inhibit igf-1r and stat3 signaling pathways in tme cancer cells and stromal cells, resulting in decreased cancer cell survival.
HC-056456;化合物HC-056456HC 056456|||3,4-Bis(2-thienoyl)-1,2,5-oxadiazole-N-oxide;HC 056456|||3,4-Bis(2 (2024/9/8)
簡介:hc-056456 (3,4-bis(2-thienoyl)-1,2,5-oxadiazole-n-oxide) is a catsper channel modulator.
PEO-IAA化合物PEO-IAA2-(1H-Indol-3-yl)-4-oxo-4-phenyl-butyric acid (2024/9/8)
簡介:peo-iaa (2-(1h-indol-3-yl)-4-oxo-4-phenyl-butyric acid) is a novel potent auxin antagonist.
Hydrocortisone hemisuccinate;氫化可的松琥珀酸酯Hydrocortisone 21-he|||hydrocortisone 21-hemisuccinate*free ac (2024/9/8)
簡介:hydrocortisone hemisuccinate (hydrocortisone 21-hemisuccinate*free acid) is a corticosteroid used as an analytical and chromatography reagent.
9-Methoxycanthin-6-one;9-甲氧基鐵屎米酮9-Methoxycanthin-6-one (2024/9/8)
簡介:9-methoxycanthin-6-one has anti-tumour activity, exhibits cytotoxic activity towards kb, lu-1, lncap, hl-60 cancer cells and other human cancer cell lines with ic50 values around 1-4 μg/ml.
BMS-3;化合物BMS3BMS-3 (2024/9/8)
簡介:bms-3 is a potent limk inhibitor with ic50s of 5 nm and 6 nm for limk1 and limk2, respectively.
HG-9-91-01;化合物HG-9-91-01SIK inhibitor 1;SIK inhibitor 1 (2024/9/8)
簡介:hg-9-91-01 (sik inhibitor 1) is a potent and highly selective salt-inducible kinase (siks) inhibitor with ic50s of 0.92 nm, 6.6 nm and 9.6 nm for sik1, sik2 and sik3respectively.
BMS-5;化合物BMS5BMS5|||LIMKi 3;BMS5|||LIMKi 3 (2024/9/8)
簡介:bms-5 (limki 3) is a potent limk inhibitor with ic50s of 7 nm and 8 nm for limk1 and limk2, respectively.
UM-164;化合物UM-164UM164|||DAS-DFGO-II;UM164|||DAS-DFGO-II (2024/9/8)
簡介:um-164 (das-dfgo-ii), a highly potent c-src inhibitor with a dissociation constant (kd) of 2.7 nm, also effectively inhibits p38α and p38β.
4-IBP;化合物4-IBP4-IBP (2024/9/8)
簡介:4-ibp is a selective σ1 agonist with a high level of affinity for the σ1 receptor (ki = 1.7 nm) and a moderate affinity for the σ2 receptor (ki = 25.2 nm) .
YHO-13177;化合物YHO-13177YHO 13177|||YHO13177;YHO 13177|||YHO13177 (2024/9/8)
簡介:yho-13177 is a potent and specific inhibitor of bcrp; potentiated the cytotoxicity of sn-38 in cancer cells and no effect on p-glycoprotein–mediated paclitaxel resistance in mdr1-transduced human leukemia k562 cells.
SR1078;化合物SR 1078SR 1078;SR 1078 (2024/9/8)
簡介:sr1078 is an agonist of retinoic acid receptor-related orphan receptor (ror)α/γ.
簡介:isopimpinellin (4,9-dimethoxypsoralen) is a natural product isolated from the roots of pimpinella saxifrage with antiviral and antileishmanial activity.
TOMATIDINE HYDROCHLORIDE鹽酸番茄堿Tomatidine|||Tomatidine HCl|||鹽酸番茄堿 (2024/9/8)
簡介:tomatidine hydrochloride (tomatidine hcl) is a steriodal alkaloid structurally similar to cyclopamine but does not inhibit hedgehog pathway. may be used as a negative control for cyclopamine and kaad-cyclopamine. tomatidine protects against muscle atrophy and boosting muscle growth.
Dihydrokavain;二氫醉椒素Marindinin|||7,8-Dihydrokavain|||7,8-Dihydrokawain;Marindinin|||二氫醉椒素|||7,8-Dihyd (2024/9/8)
簡介:dihydrokavain (marindinin), a prominent kavalactone in the kava plant, significantly contributes to the plant´s anxiolytic effects, as evidenced by a study conducted on chicks.
(+)-Kavain醉椒素醉椒素|||Kavain|||L-KAWAIN|||(R)-KAWAIN (2024/9/8)
簡介:(+)-kavain ((r)-kawain) is one of the six major kavalactones found in the piper methysticum (kava) plant; reversible inhibitor of mao-b.
Glycochenodeoxycholic Acid;甘氨鵝脫氧膽酸Glycine chenodeoxycholate|||Chenodeoxycholylglycine|||GCDCA|||Glyc (2024/9/8)
簡介:glycochenodeoxycholic acid (lithocholylglycine) is a glycine conjugate of lithocholic acid, a bile acid. it is increased in livers of mice that are fed diets supplemented with ursadeoxycholic acid. glycolithocholic acid levels are decreased in lean mice treated with obestatin. serum glycolithocholic acid levels increase with age in children.
Mirificin;芹糖葛根素苷BCP10902|||Puerarin Apioside;BCP10902|||Puerarin Apioside|||葛根素芹菜糖苷|||芹糖葛根素苷 (2024/9/8)
簡介:mirificin (bcp10902) is an active ingredient in tongmai formula (tmf) which is a well-known chinese medicinal preparation. anti-oxidant.
(Rac)-Arnebin 1;β,β-二甲基丙烯酰阿卡寧beta, beta-dimethylacrylshikonin;β,β-二甲基丙烯酰阿卡寧|||beta, beta-dimethylacr (2024/9/8)
簡介:(rac)-arnebin 1 (beta, beta-dimethylacrylshikonin) has anti-tumor, anti-inflammatory, anti-immune deficiency and protecting liver.
EGTA;乙二醇雙(2-氨基乙基醚)四乙酸Ethylenebis(oxyethylenenitrilo)tetraacet;Ethylenebis(oxyethylenenitrilo)tetraac (2024/9/8)
簡介:ethylenebis(oxyethylenenitrilo)tetraacet is a diether that is ethylene glycol in which the hydrogens of the hydroxy groups have been replaced by 2-[bis(carboxymethyl)amino]ethyl group respectively.
BMS-813160;化合物BMS813160BMS 813160;BMS 813160 (2024/9/8)
簡介:bms-813160 is the first dual ccr2/ccr5 antagonist to enter clinical development for cardiovascular.
PFI-2 hydrochloride;化合物(R)-PFI-2 hydrochloride(R)-PFI-2 hydrochloride|||PFI-2 HCl;(R)-PFI-2 hydrochl (2024/9/8)
簡介:pfi-2 hydrochloride ((r)-pfi-2 hydrochloride) is a potent, highly selective, and cell-active inhibitor of the methyltransferase activity of setd7 (ic50: 2 nm), 500 fold active than (s)-pfi-2.