9月
TP-3654；化合物TP3654TP-3654 (2024/9/8)
簡介：tp-3654 is a second-generation pim kinase inhibitor (ki values against pim-1/3: 5/42 nm).
SSD114 HCl；化合物SSD114 hydrochlorideSSD114 HCl (2024/9/8)
簡介：ssd114 is a novel gabab receptor positive allosteric modulator.
Edg-2 receptor inhibitor 1；化合物Edg-2 receptor inhibitor 1SAR-100842；SAR-100842 (2024/9/8)
簡介：edg-2 receptor inhibitor 1 (sar-100842) is an edg-2 receptor inhibitor extracted (ic50: <0.1 μm).
Berberine chloride (hydrate)化合物 T4520Natural Yellow 18 chloride hydrate|||鹽酸小檗堿水合物 (2024/9/8)
簡介：berberine chloride (hydrate) is an alkaloid from hydrastis canadensis l., berberidaceae and also found in many other plants. it is relatively toxic to parenterally but has been used orally for various fungal and parasitic infections and an anti-diarrheal.
Alisol A；澤瀉醇 AAlisol-A；Alisol-A|||澤瀉醇 A (2024/9/8)
簡介：alisol a (alisol-a) may be an autophagic inducer, it has anti-cancer activity, it presents inhibitory effects on cancer cell lines tested(hepg2, mda-mb-231, and mcf-7 cells).
Licochalcone D；甘草查爾酮 DLicochalcone D (2024/9/8)
簡介：licochalcone d may be a potential drug for human melanoma treatment by inhibiting proliferation, inducing apoptosis via the mitochondrial pathway and blocking cell migration and invasion. licochalcone d has cardioprotective potential against myocardial ischemia/reperfusion injury in langendorff-perfused rat hearts. licochalcone d has anti-inflammatory activity, it shows suppression ability of nitric oxide (no) production. licochalcone d has anti-allergic activity, it suppresses degranulation by
L189；化合物L189L189 (2024/9/8)
簡介：l189 is a human dna ligase inhibitor, inhibits hligi/iii/iv (ic50: 5/9/5 μm).
Sitsirikine；化合物 T4516Sitsirikine (2024/9/8)
簡介：sitsirikine is a natural product from catharanthus roseus.
A939572；化合物A939572A939572 (2024/9/8)
簡介：a939572 is stearoyl-coa desaturase1 (scd1) inhibitor with ic50 values of <4 nm for mscd1 and 37 nm for hscd1.
N-Acetyl-D-Glucosamine；N-乙酰-D-氨基葡萄糖NAG|||N-Acetyl-2-amino-2-deoxyglucose|||Marine Sweet|||N-Acetyl-2 (2024/9/8)
簡介：n-acetyl-d-glucosamine (nag) is a monosaccharide derivative of glucose. it is released by the action of o-glcnacase, in mammalian systems from proteins that have been post-translationally modified with o-glcnac.
Vanillyl butyl ether；香草醇丁醚4-(Butoxymethyl)-2-methoxyphenol|||Butyl vanillyl ether；4-(Butoxymethyl)-2 (2024/9/8)
簡介：vanillyl butyl ether (butyl vanillyl ether) (vbe)is a capsaicin analogue,induce sensory irritation in humans,vanillyl butyl ether is an alkoxy-substituted benzyl derivative mainly used as a flavoring agent.
Magnesium glycinate甘氨酸鎂magnesium 2-aminoacetate|||Magnesium diglycinate|||甘氨酸鎂 (2024/9/8)
簡介：magnesium glycinate (magnesium 2-aminoacetate) is a supplement that boost magnesium levels in people with a deficiency of the mineral. magnesium is a vital nutrient for regulating many body processes, including muscle and nerve function, blood sugar levels, and blood pressure. this mineral also supports the making of protein, bone, and dna.
ST271；化合物ST 271ST 271；ST 271 (2024/9/8)
簡介：st271 is an effective protein tyrosine kinase (ptk) inhibitor.
Polaprezinc；聚普瑞鋅Zinc L-carnosine；Zinc L-carnosine|||聚普瑞鋅|||L-肌肽鋅 (2024/9/8)
簡介：polaprezinc is an bioavailable chelate comprised of zinc and l-carnosine, known for its gastrointestinal protective properties, as well as its anti-ulcer, antioxidant, and anti-inflammatory effects.
Inositol nicotinate；肌醇煙酸酯Inositol niacinate|||Hexanicotol|||Myo-Inositol hexanicotinate|||Mesotal||| (2024/9/8)
簡介：inositol nicotinate (mesotal) has the effect of lowering cholesterol and expanding peripheral blood vessels for hypercholesterolemia and atherosclerosis.
Glycyl-L-Histidyl-L-Lysine；甘氨酰-L-組氨酰-L-賴氨酸Glycyl-L-Histidyl-L-Lysine (2024/9/8)
簡介：glycyl-l-histidyl-l-lysine is a liver cell growth factor and an asynthetic hepatotrophic agent that stimulates hepatic erythropoietic factor production.
Chlorphenesin；氯苯甘醚Adermykon|||Chlorophenesin|||Gecophen；Adermykon|||Chlorophenesin|||Gecophen|||氯苯甘醚 (2024/9/8)
簡介：chlorphenesin (chlorophenesin) is an antigen-associated immunosuppressant that inhibits ige-mediated histamine release. it is also used as an antimycotic agent.
Gadopentetate dimeglumine；釓噴酸葡胺Meglumine gadopentetate|||SH-L-451A|||Gd-DTPA|||Gadopentetic acid dim (2024/9/8)
簡介：gadopentetate dimeglumine (gd-dtpa), an extracellular intravenous contrast agent, is used in combination with magnetic resonance imaging (mri) to allow blood vessels, organs, and other non-bony tissues to be seen more clearly on the mri.
Ferrous Bisglycinate；甘氨酸亞鐵Bisglycine iron(II) salt|||Iron(II) bisglycinate；Bisglycine iron(II) salt| (2024/9/8)
簡介：ferrous bisglycinate (bisglycine iron(ii) salt) is used in the fortification of infant formulations and foods.
Triclocarban；三氯卡班Solubacter|||Cutisan|||Procutene|||3,4,4′-Trichlorocarbanilide；Solubacter|||Cutisan (2024/9/8)
簡介：triclocarban (cutisan), an antimicrobial agent, is used in personal cleaning products.
Talniflumate；他尼氟酯Somalgen；Somalgen|||他尼氟酯 (2024/9/8)
簡介：talniflumate (somalgen) is a calcium-activated chloride channel (hclca1/mclca3) blocker that reduces mucin synthesis and releases in animal models and cell culture. it possesses anti-inflammatory actions via inhibition of cox (cyclooxygenase) and inhibits cl-/hco3- exchange activity. it also increases survival in a cystic fibrosis mouse model of the distal intestinal obstructive syndrome.
BISMUTH SUBGALLATE次沒食子酸鉍次沒食子酸鉍|||Dermatol Puder|||Bismuth Gallate (2024/9/8)
簡介：bismuth subgallate (dermatol puder) is an astringent and antiseptic and is applied to skin diseases such as eczema.
Ceftizoxime頭孢唑肟頭孢唑肟|||Epocelin (2024/9/8)
簡介：ceftizoxime (epocelin) is a cephalosporin-based, potent antibacterial agent which can be administered intravenously or by suppository. it is highly resistant to a broad spectrum of beta-lactamases and is active against a wide range of both aerobic and anaerobic gram-positive and gram-negative organisms.
ADX88178；化合物ADX88178ADX88178 (2024/9/8)
簡介：adx88178 is a potent positive allosteric modulator for metabotropic glutamate receptor 4 (mglur4) with ec50 of 4 nm for human mglur4.
Mequitazine；美喹他嗪Metaplexan|||Virginan|||Primalan|||LM-209；Metaplexan|||Virginan|||Primalan|||LM-209| (2024/9/8)
簡介：mequitazine (virginan) is an effective, nonsedative and long-acting histamine h1 antagonist.
Stiripentol斯利潘托斯利潘托|||BCX2600|||Diacomit (2024/9/8)
簡介：stiripentol (bcx2600) (stp) is an anticonvulsant agent, which can inhibit n-demethylation of clb to nclb mediated by cyp3a4 (noncompetitively) and cyp2c19 (competitively) with ki of 1.59/0.516 μm and ic50 of 1.58/3.29 μm, respectively.
Amifampridine phosphate；化合物 T4497LBRN0110232|||3,6-DAP|||SC10|||BRN 0110232|||BRN-0110232|||NSC 5217 (2024/9/8)
簡介：amifampridine is mainly used to treat many rare muscle diseases. in the united states, aminopyridine is being studied for the treatment of lambert-eaton myasmus syndrome (lems). amifampridine is also used to treat many congenital myasthenia syndromes, particularly those with defects in choline acetyltransferase, downstream kinase 7, and any type of defects leading to "fast track" defects.
Amifampridine；阿米吡啶3,4-Pyridinediamine|||Pyridine-3,4-Diamine|||3,4-Diaminopyridine；3,4-Pyridinediami (2024/9/8)
簡介：amifampridine (3,4-diaminopyridine) is predominantly in the treatment of a number of rare muscle diseases. amifampridine works by blocking potassium channel efflux in nerve terminals so that action potential duration is increased. ca2+ channels can then be open for a longer time and allow greater acetylcholine release to stimulate muscle at the end plate.
LM22B-10；化合物LM22B-10LM22B10；LM22B10 (2024/9/8)
簡介：lm22b-10 is an activator of trkb/trkc neurotrophin receptor and can induce trkb, trkc, erk and akt activation in vitro and in vivo.
dBET1；化合物dBET1dBET1 (2024/9/8)
簡介：dbet1 is a hybrid molecule that combines (+)-jq1 and thalidomide. it induces cereblon-dependent bet protein degradation in vitro (ec50: 430 nm) and induces apoptosis.
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